Product Description INTERMEDIATES FOR PHARMACEUTICALS
No. Product Application
1. 5-acetyl-3-chloroiminodibenzyl chlomipramine hcl
2. 1-acetyl-4-(4-hydroxyphenyl)-piperazine ketonazole
3. 2-amino-5-chloro-2'-fluorobenzophenone fludiazepam
4. 2-amino-5-mercapto-1,3,4-thiadiazole acetazolamide
5. 4-amino-3,5-dichloroacetophenone clenbuterol
6. 2-apichloro-triphenylmethane clotrimazole
7. amygdalinic acid ethyl ester pemoline
8. 4-bromo-2-fluoroaniline flurbiprofen
9. 2-chloro-9-(3-dimethyl-aminopropyl)-9-hydroxy-thiox-anthene tardan
10. 2-chloro-6,7-dimethoxy-4-quinazolinamine doxazosine
11. 3-chloro-1-(4-fluorobenzenoxyl) propane sixapiride
12. 2-chloromethyl-3,5-dimethyl-4-methoxy pyridine hydrochloride omeprazole
13. chloro-phenyl-acyl-phene-oxy-isobutyric acid fenofibrate
14. 4-chloro-3-sulfamoyl benzoic acid imdapamide
15. 2-chlorothiox-anthone tartan
16. 4-(4-chlorophenyl)-4-hydroxy piperidine haloperidol
17. cyclopentanodumide gliclazide
18. cysteamin beta-hydrogenchloride famotidine
19. 2,4-dichloro-5-sulfamoyl benzoic acid furosemide
20. 1,3-dichloro-5-sulfamoyl benzoic acid amikacin
21. 3-(3,4-dimethoxyphenyl) acetone methyldoba
22. dimethyl N-cyanodithioiminocarbonate ranitidine
23. 6,7-dimethyloxy-2,4-(1H,3H) quinazoline dione doxazosine
24. diphenyl ketone clonazepam
25. diphenyl acetonitrile doxaram
26. dl-naproxen naproxen
27. 4-fluoro benzylamine azmizole
28. 2-fluoro-4-bromobiphenyl flurbirofen
29. guanine acyclovir
30. 4-hydroxy-4'-chlorobenzophen procetofen
31. 4-methyl-4-hydroxy-2H-1,2-benzothiazine-3-carboxylic acid ethylester-1,1-dioxide piraxicam
32. 2-methyl-1,4-naphthoquinone vitamin k3
33. 2-nitrobenzaldehyde nifedipine
34. 4-anisidine andipine
35. 4-chloromethylbenzoic acid tranexamic acid
36. 4-hydroxyphenyl acetamide atinolol
37. 4-phenexidine ophenacedine
38. 4-toluic acid tranexamic aci
39. 1,1,3-trichloroacetone folic acid
40. 1-(1H-2,4-trizole-1-)-2-(2,4-diflubenzen)-aceton fluconazole
41. piperacillin free acid piperacillin+tazobactam
42. tazobactam free acid piperacillin+tazobactam
43. sulbactam free acid ampicillin+sulbactam
44. penicillin G salt
ANTIBIOTIC INTERMEDIATES
A. SIDE CHAINS FOR CEPHALOSPORIN PRODUCTS
1. HO-EPCP=D-(-)-2-[(4-Ethyl-2,3-Dioxo-1-Peperazineyl)-Carbonylamino]-2-(4-Hydroxyphenyl) Acetic Acid
2. MMTZ=1-Methyl-5-Mercapto-1,2,3,4-Tetrazole
3. SMIA(AMF)=(Z)-2-Methoxyimino-(Furyl-2-yl) Acetic Acid Ammonium Salt
4. MTD=2-Mercapto-1,3,4-Thiadiazole
5. AMAA=(Z)-2-Methoxyimino-2-(2-Aminothiazol-4-yl) Acetic Acid Anhydrous
6. MAEM=(Benzothiazol-2-yl)-2-(2-Aminothiazol-4-yl)-(Z)-2-Methoxyimino Thioacetate
7. EHATA=Ethyl-(Z)-2-Hydroxyimino-2-(2-Aminothiazol-4-yl) Acetate
8. HATA=(Z)-2-Hydroxyimino-2-(2-Aminothiazol-4-yl) Acetic Acid
9. EATA=Ethyl-2-(2-Aminothiazole-4-yl) Acetate
10. ATAA=2-(2-Aminothiazol-4-yl) Acetic Acid
11. AT-TBA=(Z)-2-(Tert-Butoxycarbonylprop-2-Oxyimino)-2-(2-Aminothiazol-4-yl) Acetic Acid
12. BPTA=Benzothiazol-yl-(Z)-2-(Tert-Butoxycarbonylprop-2-Oxyimino)-2-(2-Aminothiazol-4-yl)
Thioacetate
13. SMT=5-Mercapto-1,2,3,4-Tetrazole-1-Methyl Sulfonic Acid
14. SMT-DS=5-Mercapto-1,2,3,4-Tetrazole-1-Methyl Sulfonic Acid Disodium Salt
15. TAC=Thiophene-2-Actyl Chloride
16. PG=D-(-)Phenylglycine
17. PGDS=D-(-)Phenylglycine Dane Salt
18. PG-AMIDE=D-(-)Phenyglycine Amide
19. PG-CL=D-(-)Phenylglycinic Chloride
20. DHPG=D-(-) Dihydro Phenylglycine Base
21. DIPGDS=D-(-)Dihydro Phenylglycine Dane Salt
22. TAA=1H-Tetrazolyl-1-Acetic Acid
23. MMTD=2-Mercapto-5-Methyl-1,3,4-Thiadiazole
B. INTERMEDIATES FOR QUINOLINE
1) 1-Ethyl-6-Fluoro-7-Chloro-1,4-Dihydro-4-Oxo-3-Quinolinecarxylic Acid For Norfloxacin
2) 9-Fluoro-2,3-Dihydro-3-Methyl-10-Chloro-7-7H-Pyrido(1,2,3-de)-1,4-Benzoxazine-6-Carboxylic Acid For Ofloxacin
3) 1-Cyclopropyl-6-Fluoro-7-Chloro-1,4-Dihydro-4-Oxo-3-Quinolinecarboxylic Acid For
Ciprofloxacin
4) 1-Ethy-6-Fluoro-7-Chloro-1,4-Dihydro-4-Oxo-1,8-Naphthylidine-3-Carbonxylic Acid For
Enoxacin
5) 1-Cyclopropyl-6-Fluoro-7-Chloro-1,4-Dihydro-4-Oxo-1,8-Naphthylidine-3-Carboxylic Acid
For New Quinoline
6) Levofloxacin Carboxylic Acid For Levofloxacin
7) L-alaninol For Levofloxacin
8) 1-Ethyl-6,7,8-Trifluoro-1,4-Dihydro-4-Oxo-Quinoline-3-Carboxylic Acid For Lomefloxacin
9) 1-Acetone-Oxo-3,4-Difluoro-Nitrobenzene For Ofloxacin
antibiotics
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